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Описание

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Клотримазол крем д/нар. прим., 1%, 20 г

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Коротко о товаре

Артикул Маркета
2101370425737
Действующее вещество
Форма выпуска
крем
Инструкция
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Крем следует наносить на пораженные участки кожи 2-3 раза/сут.\u003Cbr\u003EДля профилактики рецидивов лечение следует продолжать, по крайней мере, в течение двух недель после исчезновения всех симптомов инфекции.\u003Cbr\u003EКрем следует наносить на чистые сухие участки пораженной кожи (вымытой мылом с нейтральным рН), на стопы крем следует наносить между пальцами.\u003Cbr\u003EПродолжительность лечения зависит тяжести заболевания, его локализации, эффективности лечения.\u003Cbr\u003EПродолжительность лечения: дерматомикозы - 3-4 недели; эритразма - 2-4 недели; разноцветный лишай - 1-3 недели; кандидозный вульвит и баланит - 1-2 недели.\u003Cbr\u003EПродолжительность лечения может меняться в соответствии с индивидуальными особенностями, но не рекомендуется продолжительность лечения менее 3 недель. Для профилактики рецидивов инфекции следует продолжать применение препарата в течение 1-2 недель после исчезновения всех симптомов заболевания. Если после 7 дней лечения не наступает улучшение симптоматики, необходимо проконсультироваться с врачом."},{"name":"Побочные действия","value":"Нежелательные явления, представленные ниже, перечислены в соответствии с поражением органов и систем органов и частотой встречаемости. Частота встречаемости определяется следующим образом: очень часто (≥1/10), часто (≥1/100 и \u003C 1/10), нечасто (≥1/1000 и \u003C 1/100), редко (≥1/10 000 и \u003C 1/1 000), очень редко (\u003C 1/10 000, включая отдельные случаи), неизвестно (частота не может быть оценена по имеющимся на настоящий момент данным). Категории частоты были сформированы на основании пострегистрационного наблюдения.\u003Cbr\u003EСо стороны иммунной системы: неизвестно - аллергическая реакция (проявляющаяся крапивницей, обмороком, артериальной гипотензией, одышкой).\u003Cbr\u003EСо стороны кожи и подкожных тканей: неизвестно - сыпь, зуд, пузырьковые высыпания, шелушение, боль или дискомфорт, отек, жжение, раздражение."},{"name":"Фармакологическое действие","value":"Клотримазол подавляет рост и деление микроорганизмов и, в зависимости концентрации, может оказывать фунгистатическое (задерживающее и останавливающее рост клеток грибов) или фунгицидное (приводящее к гибели грибов) действие. Клотримазол угнетает синтез эргостерола и связывается с фосфолипидами клеточной мембраны гриба, что приводит к изменению проницаемости мембран клеток.\u003Cbr\u003EВ более высоких концентрациях клотримазол вызывает повреждение клеточных мембран по механизмам, не зависящим синтеза стеролов.\u003Cbr\u003EКлотримазол также нарушает процессы жизнедеятельности в клетке гриба, подавляя образование компонентов, необходимых для построения жизненно-важных клеточных структур (белков, жиров, ДНК, полисахаридов), повреждает нуклеиновые кислоты и увеличивает выведение калия.\u003Cbr\u003EВ конечном итоге воздействие клотримазола на грибковые клетки приводит к их гибели.\u003Cbr\u003EКлотримазол характеризуется широким спектром противогрибковой и антибактериальной активности: дерматофиты (Epidermophyton floccosum, Microsporum canis, Trichophyton mentagrophytes, Trichophyton rubrum), дрожжи (Candida spp., Cryptococcus neoformans), диморфные грибы (Coccidioides immitis, Histoplasma capsulatum, Paracoccidioides brasiliensis), простейшие (Trichomonas vaginalis).\u003Cbr\u003EТакже он активен в отношении некоторых грамположительных бактерий.\u003Cbr\u003EПри изучении эффективности клотримазола в лабораторных условиях вне организма человека (in vitro) выявлен широкий спектр его фунгистатической и фунгицидной активности. Он воздействует на мицелий дерматофитов (Trichophyton, Microsporum, Epidermophyton) аналогично гризеофульвину, а его действие на почкующиеся грибы (Candida) аналогично действию полиенов (амфотерицина В и нистатина).\u003Cbr\u003EВ концентрациях менее 1 мкг/мл клотримазол подавляет развитие большинства штаммов болезнетворных грибов, относящихся к Trichophyton rubrum, Trichophyton mentagrophytes, Epidermophyton floccosum, Microsporum canis.\u003Cbr\u003EВ концентрации 3 мкг/мл клотримазол подавляет развитие большинства других бактерий: Pityrosporum orbiculare, Aspergillus fumigatus, рода Candida, в т.ч. Candida albicans, некоторых штаммов Staphylococcus aureus, Streptococcus pyogenes, а также некоторых штаммов Proteus vulgaris и Salmonella. Клотримазол активен в отношении Sporothrix, Cryptococcus, Cephalosporium, Fusarium.\u003Cbr\u003EВ концентрациях более 100 мкг/мл он эффективен в отношении Trichomonas vaginalis.\u003Cbr\u003EГрибы, устойчивые к клотримазолу, встречаются крайне редко; есть данные только по отдельным штаммам Candida guilliermondii.\u003Cbr\u003EНе сообщалось о развитии устойчивости у чувствительных к клотримазолу грибов после пассажа Candida albicans и Trichophyton mentagrophytes. Не описано случаев развития устойчивости к клотримазолу у штаммов Candida albicans, устойчивых к полиеновым антибиотикам вследствие химической мутации."},{"name":"Фармакологическая группа","value":"противогрибковые средства"},{"name":"Форма выпуска","value":"крем"},{"name":"Способ применения/введения","value":"наружный","transition":{"type":"catalog","params":{"categorySlug":"sredstva-ot-gribka","categoryId":"15756513","navnodeId":"72474","glfilters":["35947170:36763741"]}}},{"name":"Условия хранения","value":"Препарат следует в недоступном для детей месте при температуре не выше 25 ° С. Не замораживать. Срок годности - 3 года."},{"name":"Передозировка","value":"Симптомы: при случайном приеме препарата внутрь возможно появление головокружения, тошноты, рвоты.\u003Cbr\u003EЛечение: при случайном приеме крема внутрь следует проводить симптоматическое лечение. При наружном применении препарата передозировка маловероятна."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Не сообщалось о влиянии клотримазола на способность управлять транспортными средствами и механизмами."},{"name":"Особые указания","value":"Необходимо избегать попадания крема на слизистую оболочку глаз. Не глотать.\u003Cbr\u003EВсе инфицированные области следует лечить одновременно.\u003Cbr\u003EВ состав препарата Клотримазол входит цетостеариловый спирт, который может вызывать местные кожные реакции (например, контактный дерматит).\u003Cbr\u003EПри появлении симптомов повышенной чувствительности или раздражения лечение прекращают.\u003Cbr\u003EДанные лабораторных исследований свидетельствуют о том, что использование контрацептивов, содержащих латекс, может вызывать их повреждение при совместном применении с клотримазолом. Следовательно, эффективность таких контрацептивов может снижаться. Пациентам следует рекомендовать применение альтернативных методов контрацепции в течение, по крайней мере, 5 дней после применения клотримазола."},{"name":"Взаимодействие","value":"Не изучалось."},{"name":"Регистрационный номер","value":"П N011413/02"},{"name":"Дата государственной регистрации","value":"12.12.2018"},{"name":"Владелец регистрационного удостоверения","value":"GlaxoSmithKline","transition":{"type":"catalog","params":{"categorySlug":"sredstva-ot-gribka","categoryId":"15756513","navnodeId":"72474","glfilters":["34324371:35649313","7893318:11906905"]}}},{"name":"Изготовитель","value":"GlaxoSmithKline"},{"name":"Фасовщик","value":"GlaxoSmithKline"},{"name":"Страна бренда","value":"Великобритания"},{"name":"Страна-производитель","value":"Польша"},{"name":"Название препарата","value":"Клотримазол","transition":{"type":"catalog","params":{"categorySlug":"sredstva-ot-gribka","categoryId":"15756513","navnodeId":"72474","glfilters":["17796364:17876928"]}}},{"name":"Срок годности","value":"36 мес."}]}},"fullSpecsGrouped":{"9904639783257658855":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Органы и системы","value":"кожа"},{"name":"Назначение","value":"грибок кожи, микоз стоп, разноцветный лишай"},{"name":"Показания к применению","value":"Для наружного лечения грибковых заболеваний кожи, вызванных дерматофитами, дрожжеподобными грибами, плесневыми грибами, а также возбудителями, чувствительными к клотримазолу:\u003Cbr\u003Eмикозы стоп, кистей, туловища, кожных складок;\u003Cbr\u003Eкандидозный вульвит, кандидозный баланит;\u003Cbr\u003Eразноцветный лишай, эритразма;\u003Cbr\u003Eгрибковые инфекции наружного уха."},{"name":"Противопоказания","value":"Повышенная чувствительность к клотримазолу или другим компонентам препарата."},{"name":"Состав","value":"Действующее вещество: клотримазол – 1 г.\u003Cbr\u003EВспомогательные вещества: бензиловый спирт – 1 г, цетостеариловый спирт – 11.5 г, октилдодеканол – 10 г, полисорбат 60 – 1.5 г, сорбитан стеарат – 2 г, спермацет синтетический – 3 г, вода – 71 г (вводят с избытком 1.5%, который удаляется по ходу технологического процесса).\u003Cbr/\u003E"},{"name":"Действующее вещество","value":"Клотримазол"},{"name":"Способ применения и дозы","value":"Для наружного применения. Крем следует наносить на пораженные участки кожи 2-3 раза/сут.\u003Cbr\u003EДля профилактики рецидивов лечение следует продолжать, по крайней мере, в течение двух недель после исчезновения всех симптомов инфекции.\u003Cbr\u003EКрем следует наносить на чистые сухие участки пораженной кожи (вымытой мылом с нейтральным рН), на стопы крем следует наносить между пальцами.\u003Cbr\u003EПродолжительность лечения зависит тяжести заболевания, его локализации, эффективности лечения.\u003Cbr\u003EПродолжительность лечения: дерматомикозы - 3-4 недели; эритразма - 2-4 недели; разноцветный лишай - 1-3 недели; кандидозный вульвит и баланит - 1-2 недели.\u003Cbr\u003EПродолжительность лечения может меняться в соответствии с индивидуальными особенностями, но не рекомендуется продолжительность лечения менее 3 недель. Для профилактики рецидивов инфекции следует продолжать применение препарата в течение 1-2 недель после исчезновения всех симптомов заболевания. Если после 7 дней лечения не наступает улучшение симптоматики, необходимо проконсультироваться с врачом."},{"name":"Побочные действия","value":"Нежелательные явления, представленные ниже, перечислены в соответствии с поражением органов и систем органов и частотой встречаемости. Частота встречаемости определяется следующим образом: очень часто (≥1/10), часто (≥1/100 и \u003C 1/10), нечасто (≥1/1000 и \u003C 1/100), редко (≥1/10 000 и \u003C 1/1 000), очень редко (\u003C 1/10 000, включая отдельные случаи), неизвестно (частота не может быть оценена по имеющимся на настоящий момент данным). Категории частоты были сформированы на основании пострегистрационного наблюдения.\u003Cbr\u003EСо стороны иммунной системы: неизвестно - аллергическая реакция (проявляющаяся крапивницей, обмороком, артериальной гипотензией, одышкой).\u003Cbr\u003EСо стороны кожи и подкожных тканей: неизвестно - сыпь, зуд, пузырьковые высыпания, шелушение, боль или дискомфорт, отек, жжение, раздражение."},{"name":"Фармакологическое действие","value":"Клотримазол подавляет рост и деление микроорганизмов и, в зависимости концентрации, может оказывать фунгистатическое (задерживающее и останавливающее рост клеток грибов) или фунгицидное (приводящее к гибели грибов) действие. Клотримазол угнетает синтез эргостерола и связывается с фосфолипидами клеточной мембраны гриба, что приводит к изменению проницаемости мембран клеток.\u003Cbr\u003EВ более высоких концентрациях клотримазол вызывает повреждение клеточных мембран по механизмам, не зависящим синтеза стеролов.\u003Cbr\u003EКлотримазол также нарушает процессы жизнедеятельности в клетке гриба, подавляя образование компонентов, необходимых для построения жизненно-важных клеточных структур (белков, жиров, ДНК, полисахаридов), повреждает нуклеиновые кислоты и увеличивает выведение калия.\u003Cbr\u003EВ конечном итоге воздействие клотримазола на грибковые клетки приводит к их гибели.\u003Cbr\u003EКлотримазол характеризуется широким спектром противогрибковой и антибактериальной активности: дерматофиты (Epidermophyton floccosum, Microsporum canis, Trichophyton mentagrophytes, Trichophyton rubrum), дрожжи (Candida spp., Cryptococcus neoformans), диморфные грибы (Coccidioides immitis, Histoplasma capsulatum, Paracoccidioides brasiliensis), простейшие (Trichomonas vaginalis).\u003Cbr\u003EТакже он активен в отношении некоторых грамположительных бактерий.\u003Cbr\u003EПри изучении эффективности клотримазола в лабораторных условиях вне организма человека (in vitro) выявлен широкий спектр его фунгистатической и фунгицидной активности. Он воздействует на мицелий дерматофитов (Trichophyton, Microsporum, Epidermophyton) аналогично гризеофульвину, а его действие на почкующиеся грибы (Candida) аналогично действию полиенов (амфотерицина В и нистатина).\u003Cbr\u003EВ концентрациях менее 1 мкг/мл клотримазол подавляет развитие большинства штаммов болезнетворных грибов, относящихся к Trichophyton rubrum, Trichophyton mentagrophytes, Epidermophyton floccosum, Microsporum canis.\u003Cbr\u003EВ концентрации 3 мкг/мл клотримазол подавляет развитие большинства других бактерий: Pityrosporum orbiculare, Aspergillus fumigatus, рода Candida, в т.ч. Candida albicans, некоторых штаммов Staphylococcus aureus, Streptococcus pyogenes, а также некоторых штаммов Proteus vulgaris и Salmonella. Клотримазол активен в отношении Sporothrix, Cryptococcus, Cephalosporium, Fusarium.\u003Cbr\u003EВ концентрациях более 100 мкг/мл он эффективен в отношении Trichomonas vaginalis.\u003Cbr\u003EГрибы, устойчивые к клотримазолу, встречаются крайне редко; есть данные только по отдельным штаммам Candida guilliermondii.\u003Cbr\u003EНе сообщалось о развитии устойчивости у чувствительных к клотримазолу грибов после пассажа Candida albicans и Trichophyton mentagrophytes. Не описано случаев развития устойчивости к клотримазолу у штаммов Candida albicans, устойчивых к полиеновым антибиотикам вследствие химической мутации."},{"name":"Фармакологическая группа","value":"противогрибковые средства"},{"name":"Форма выпуска","value":"крем"},{"name":"Способ применения/введения","value":"наружный"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"Препарат следует в недоступном для детей месте при температуре не выше 25 ° С. Не замораживать. Срок годности - 3 года."},{"name":"Передозировка","value":"Симптомы: при случайном приеме препарата внутрь возможно появление головокружения, тошноты, рвоты.\u003Cbr\u003EЛечение: при случайном приеме крема внутрь следует проводить симптоматическое лечение. При наружном применении препарата передозировка маловероятна."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Не сообщалось о влиянии клотримазола на способность управлять транспортными средствами и механизмами."},{"name":"Особые указания","value":"Необходимо избегать попадания крема на слизистую оболочку глаз. Не глотать.\u003Cbr\u003EВсе инфицированные области следует лечить одновременно.\u003Cbr\u003EВ состав препарата Клотримазол входит цетостеариловый спирт, который может вызывать местные кожные реакции (например, контактный дерматит).\u003Cbr\u003EПри появлении симптомов повышенной чувствительности или раздражения лечение прекращают.\u003Cbr\u003EДанные лабораторных исследований свидетельствуют о том, что использование контрацептивов, содержащих латекс, может вызывать их повреждение при совместном применении с клотримазолом. Следовательно, эффективность таких контрацептивов может снижаться. Пациентам следует рекомендовать применение альтернативных методов контрацепции в течение, по крайней мере, 5 дней после применения клотримазола."},{"name":"Взаимодействие","value":"Не изучалось."},{"name":"Регистрационный номер","value":"П N011413/02"},{"name":"Дата государственной регистрации","value":"12.12.2018"},{"name":"Владелец регистрационного удостоверения","value":"GlaxoSmithKline"},{"name":"Изготовитель","value":"GlaxoSmithKline"},{"name":"Фасовщик","value":"GlaxoSmithKline"},{"name":"Страна бренда","value":"Великобритания"},{"name":"Страна-производитель","value":"Польша"},{"name":"Название препарата","value":"Клотримазол"},{"name":"Срок годности","value":"36 мес."}]}],"transitionId":"tr_12770343965740482778"}}}}
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Инструкция

Показания к применению

Для наружного лечения грибковых заболеваний кожи, вызванных дерматофитами, дрожжеподобными грибами, плесневыми грибами, а также возбудителями, чувствительными к клотримазолу:
микозы стоп, кистей, туловища, кожных складок;
кандидозный вульвит, кандидозный баланит;
разноцветный лишай, эритразма;
грибковые инфекции наружного уха.

Противопоказания

Повышенная чувствительность к клотримазолу или другим компонентам препарата.

Способ применения и дозы

Для наружного применения. Крем следует наносить на пораженные участки кожи 2-3 раза/сут.
Для профилактики рецидивов лечение следует продолжать, по крайней мере, в течение двух недель после исчезновения всех симптомов инфекции.
Крем следует наносить на чистые сухие участки пораженной кожи (вымытой мылом с нейтральным рН), на стопы крем следует наносить между пальцами.
Продолжительность лечения зависит тяжести заболевания, его локализации, эффективности лечения.
Продолжительность лечения: дерматомикозы - 3-4 недели; эритразма - 2-4 недели; разноцветный лишай - 1-3 недели; кандидозный вульвит и баланит - 1-2 недели.
Продолжительность лечения может меняться в соответствии с индивидуальными особенностями, но не рекомендуется продолжительность лечения менее 3 недель. Для профилактики рецидивов инфекции следует продолжать применение препарата в течение 1-2 недель после исчезновения всех симптомов заболевания. Если после 7 дней лечения не наступает улучшение симптоматики, необходимо проконсультироваться с врачом.
Полная инструкция
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Клотримазол крем д/нар. прим.
Клотримазол крем д/нар. прим., 1%, 20 г
У продавца: 
нет • На Маркете: 4.6
(52)
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Инструкция
Нет в продаже
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У других продавцов:52 оценки·14 отзывов
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