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Описание

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Кестин таб. лиоф., 20 мг, 10 шт.

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У продавца: 
нет • На Маркете: 4.8
(66)
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Коротко о товаре

Артикул Маркета
2186887793
Действующее вещество
Возраст
от 12 лет
Инструкция
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При недостаточной эффективности или выраженной симптоматике рекомендуется использовать препарат Кестин, таблетки лиофилизированные 20 мг, по 1 таблетке 1 раз в сутки.\u003Cbr\u003EКурс лечения будет определяться исчезновением симптомов заболевания.\u003Cbr\u003EПожилые пациенты: коррекции дозы не требуется.\u003Cbr\u003EПациенты с нарушенной функцией почек: коррекции дозы не требуется. Пациенты с легкой и умеренной печеночной недостаточностью: коррекции дозы не требуется.\u003Cbr\u003EПри тяжелых нарушениях функции печени (класс С по классификации Чайлд-Пью) суточная доза не должна превышать 10 мг, поэтому рекомендуется в этих случаях использовать препарат Кестин, таблетки, покрытые пленочной оболочкой, 10 мг.\u003Cbr\u003EИзвлечение препарата из блистера должно осуществляться сухими руками в соответствии с инструкцией ниже:\u003Cbr\u003EСпециальные предосторожности при обращении с препаратом:\u003Cbr\u003E1. Во избежание повреждения таблеток, не доставайте препарат из блистера посредством нажатия. Откройте ячейку блистера, осторожно подняв свободный край защитной пленки.\u003Cbr\u003E2. Снимите защитную пленку.\u003Cbr\u003E3. Осторожно выдавите таблетку из ячейки, не прикасаясь к ней.\u003Cbr\u003E4. Аккуратно извлеките препарат и положите его на язык, где он быстро растворится. Нет необходимости запивать водой или другой жидкостью, прием пищи не влияет на действие препарата."},{"name":"Побочные действия","value":"Ниже перечислены нежелательные реакции, наблюдавшиеся в клинических исследованиях и в ходе пострегистрационного применения препарата, с учетом следующих критериев: очень часто (≥1/10); часто (от 1/100 до \u003C1/10); нечасто (от 1/1000 до \u003C1/100); редко (от 1/10000 до \u003C 1/1000); очень редко (\u003C1/10000).\u003Cbr\u003EСо стороны центральной и периферической нервной системы:\u003Cbr\u003Eредко: сонливость;\u003Cbr\u003Eочень редко: головокружение,\u003Cbr\u003Eгипестезия, головная боль, нервозность, бессонница.\u003Cbr\u003EСо стороны желудочно-кишечного тракта:\u003Cbr\u003Eредко: сухость слизистой оболочки полости рта;\u003Cbr\u003Eочень редко: рвота, боль в животе, тошнота, диспепсия.\u003Cbr\u003EСо стороны сердечно-сосудистой системы:\u003Cbr\u003Eочень редко: сердцебиение, тахикардия.\u003Cbr\u003EСо стороны печени и желчевыводящих путей:\u003Cbr\u003Eочень редко: отклонения функциональных проб печени.\u003Cbr\u003EСо стороны кожи и подкожно-жировой клетчатки:\u003Cbr\u003Eочень редко: крапивница, сыпь, дерматит.\u003Cbr\u003EСо стороны репродуктивной системы:\u003Cbr\u003Eочень редко: менструальные расстройства.\u003Cbr\u003EОбщие и местные реакции:\u003Cbr\u003Eочень редко: отеки, астенический синдром.\u003Cbr\u003EНежелательные реакции, наблюдавшиеся в клинических исследованиях у детей старше 12 лет (группа детей из 460 человек), не отличались от реакций, отмеченных у взрослых."},{"name":"Фармакологическое действие","value":"Эбастин является блокатором Н1 -гистаминовых рецепторов длительного действия. После приема препарата внутрь выраженное противоаллергическое действие начинается через 1 ч и длится более 48 ч. После 5-дневного курса лечения препаратом Кестин антигистаминная активность сохраняется в течение 72 ч за счет действия активных метаболитов. При длительном приеме сохраняется высокий уровень блокады периферических Н1-гистаминовых рецепторов без развития тахифилаксии. Препарат не оказывает выраженного антихолинергического и седативного эффекта, не проникает через гематоэнцефалический барьер. Не отмечено влияния препарата Кестин на интервал QT на ЭКГ в дозе 100 мг - дозе, превышающей рекомендованную суточную дозу (20 мг) в 5 раз."},{"name":"Фармакологическая группа","value":"H1-антигистаминные средства"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный","transition":{"type":"catalog","params":{"categorySlug":"sredstva-ot-allergii","categoryId":"15756502","navnodeId":"72464","glfilters":["35947170:36763744"]}}},{"name":"Минимальный возраст применения","value":"от 12 лет"},{"name":"Условия хранения","value":"Хранить при температуре не выше 25 °С.\u003Cbr\u003EХранить в недоступном для детей месте."},{"name":"Передозировка","value":"В исследованиях с использованием высоких доз (более 100 мг в сутки) не наблюдалось клинически значимых признаков и симптомов. Специального антидота для эбастина нет. В случае передозировки рекомендуется промывание желудка, контроль жизненно важных функций организма, симптоматическое лечение."},{"name":"Применение при беременности и кормлении грудью","value":"Безопасность применения препарата Кестин у беременных женщин не исследована, поэтому принимать препарат во время беременности не рекомендуется.\u003Cbr\u003EКормящим матерям не рекомендуется принимать препарат Кестин, поскольку неизвестно выделяется ли эбастин с грудным молоком. При необходимости применения препарата в период лактации необходимо решить вопрос о прекращении грудного вскармливания."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"В случае возникновения побочных эффектов со стороны центральной нервной системы, таких как сонливость, необходимо соблюдать осторожность при управлении транспортными средствами и занятиях другими потенциально опасными видами деятельности, требующими повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"Эбастин может искажать результаты кожных аллергических проб. Поэтому рекомендуется проводить такие пробы не ранее, чем через 5-7 дней после отмены препарата.\u003Cbr\u003EС осторожностью:\u003Cbr\u003EПрименять у пациентов с увеличенным интервалом QT на ЭКГ, гипокалиемией, при почечной недостаточности и с легкой и умеренной степенью печеночной недостаточности (класс А, В по классификации Чайлд-Пью).\u003Cbr\u003EС осторожностью следует применять препарат Кестин при одновременном приеме с кетоконазолом или итраконазолом и эритромицином - возможно увеличение риска удлинения интервала QT на ЭКГ."},{"name":"Взаимодействие","value":"При одновременном применении препарата Кестин с кетоконазолом или итраконазолом и эритромицином возможно увеличение риска удлинения интервала QT на ЭКГ.\u003Cbr\u003EРифампицин снижает концентрацию эбастина в плазме крови и оказывает ингибирующее влияние на антигистаминный эффект эбастина.\u003Cbr\u003EПрепарат Кестин не взаимодействует с теофиллином, непрямыми антикоагулянтами, циметидином, диазепамом, этанолом и этанолсодержащими препаратами."},{"name":"Регистрационный номер","value":"ЛП-000789"},{"name":"Дата государственной регистрации","value":"14.07.2021"},{"name":"Владелец регистрационного удостоверения","value":"Almirall","transition":{"type":"catalog","params":{"categorySlug":"sredstva-ot-allergii","categoryId":"15756502","navnodeId":"72464","glfilters":["34324371:35649313","7893318:16003820"]}}},{"name":"Изготовитель","value":"Catalent U.K. Swindon Zydis Ltd"},{"name":"Фасовщик","value":"Catalent U.K. Swindon Zydis Ltd"},{"name":"Страна бренда","value":"Испания"},{"name":"Страна-производитель","value":"Великобритания"},{"name":"Название препарата","value":"Кестин","transition":{"type":"catalog","params":{"categorySlug":"sredstva-ot-allergii","categoryId":"15756502","navnodeId":"72464","glfilters":["17796364:17877896"]}}},{"name":"Срок годности","value":"36 мес."}]}},"fullSpecsGrouped":{"2074419448785158868":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Органы и системы","value":"кожа, носоглотка"},{"name":"Назначение","value":"аллергический ринит, крапивница"},{"name":"Показания к применению","value":"-аллергический ринит различной этиологии (сезонный и/или круглогодичный);\u003Cbr\u003E- крапивница различной этиологии, в том числе хроническая идиопатическая."},{"name":"Противопоказания","value":"- повышенная чувствительность к компонентам препарата;\u003Cbr\u003E- беременность;\u003Cbr\u003E- период лактации;\u003Cbr\u003E- фенилкетонурия;\u003Cbr\u003E- детский возраст до 12 лет;\u003Cbr\u003E- тяжелые нарушения функции печени (класс С по классификации Чайлд-Пью)."},{"name":"Состав","value":"1 таб.: эбастин - 20 мг.\u003Cbr\u003E\nВспомогательные вещества: магния стеарат, целлюлоза микрокристаллическая, крахмал кукурузный прежелатинизированный, лактозы моногидрат (177 мг), натрия кроскармеллоза, гипромеллоза, титана диоксид, макрогол 6000 (полиэтиленгликоль 6000)."},{"name":"Действующее вещество","value":"Эбастин"},{"name":"Способ применения и дозы","value":"Для рассасывания в полости рта, независимо от приема пищи.\u003Cbr\u003EВзрослым и детям старше 12 лет рекомендуется начинать терапию с дозы 10 мг 1 раз в сутки, используя препарат Кестин, таблетки, покрытые пленочной оболочкой, 10 мг. При недостаточной эффективности или выраженной симптоматике рекомендуется использовать препарат Кестин, таблетки лиофилизированные 20 мг, по 1 таблетке 1 раз в сутки.\u003Cbr\u003EКурс лечения будет определяться исчезновением симптомов заболевания.\u003Cbr\u003EПожилые пациенты: коррекции дозы не требуется.\u003Cbr\u003EПациенты с нарушенной функцией почек: коррекции дозы не требуется. Пациенты с легкой и умеренной печеночной недостаточностью: коррекции дозы не требуется.\u003Cbr\u003EПри тяжелых нарушениях функции печени (класс С по классификации Чайлд-Пью) суточная доза не должна превышать 10 мг, поэтому рекомендуется в этих случаях использовать препарат Кестин, таблетки, покрытые пленочной оболочкой, 10 мг.\u003Cbr\u003EИзвлечение препарата из блистера должно осуществляться сухими руками в соответствии с инструкцией ниже:\u003Cbr\u003EСпециальные предосторожности при обращении с препаратом:\u003Cbr\u003E1. Во избежание повреждения таблеток, не доставайте препарат из блистера посредством нажатия. Откройте ячейку блистера, осторожно подняв свободный край защитной пленки.\u003Cbr\u003E2. Снимите защитную пленку.\u003Cbr\u003E3. Осторожно выдавите таблетку из ячейки, не прикасаясь к ней.\u003Cbr\u003E4. Аккуратно извлеките препарат и положите его на язык, где он быстро растворится. Нет необходимости запивать водой или другой жидкостью, прием пищи не влияет на действие препарата."},{"name":"Побочные действия","value":"Ниже перечислены нежелательные реакции, наблюдавшиеся в клинических исследованиях и в ходе пострегистрационного применения препарата, с учетом следующих критериев: очень часто (≥1/10); часто (от 1/100 до \u003C1/10); нечасто (от 1/1000 до \u003C1/100); редко (от 1/10000 до \u003C 1/1000); очень редко (\u003C1/10000).\u003Cbr\u003EСо стороны центральной и периферической нервной системы:\u003Cbr\u003Eредко: сонливость;\u003Cbr\u003Eочень редко: головокружение,\u003Cbr\u003Eгипестезия, головная боль, нервозность, бессонница.\u003Cbr\u003EСо стороны желудочно-кишечного тракта:\u003Cbr\u003Eредко: сухость слизистой оболочки полости рта;\u003Cbr\u003Eочень редко: рвота, боль в животе, тошнота, диспепсия.\u003Cbr\u003EСо стороны сердечно-сосудистой системы:\u003Cbr\u003Eочень редко: сердцебиение, тахикардия.\u003Cbr\u003EСо стороны печени и желчевыводящих путей:\u003Cbr\u003Eочень редко: отклонения функциональных проб печени.\u003Cbr\u003EСо стороны кожи и подкожно-жировой клетчатки:\u003Cbr\u003Eочень редко: крапивница, сыпь, дерматит.\u003Cbr\u003EСо стороны репродуктивной системы:\u003Cbr\u003Eочень редко: менструальные расстройства.\u003Cbr\u003EОбщие и местные реакции:\u003Cbr\u003Eочень редко: отеки, астенический синдром.\u003Cbr\u003EНежелательные реакции, наблюдавшиеся в клинических исследованиях у детей старше 12 лет (группа детей из 460 человек), не отличались от реакций, отмеченных у взрослых."},{"name":"Фармакологическое действие","value":"Эбастин является блокатором Н1 -гистаминовых рецепторов длительного действия. После приема препарата внутрь выраженное противоаллергическое действие начинается через 1 ч и длится более 48 ч. После 5-дневного курса лечения препаратом Кестин антигистаминная активность сохраняется в течение 72 ч за счет действия активных метаболитов. При длительном приеме сохраняется высокий уровень блокады периферических Н1-гистаминовых рецепторов без развития тахифилаксии. Препарат не оказывает выраженного антихолинергического и седативного эффекта, не проникает через гематоэнцефалический барьер. Не отмечено влияния препарата Кестин на интервал QT на ЭКГ в дозе 100 мг - дозе, превышающей рекомендованную суточную дозу (20 мг) в 5 раз."},{"name":"Фармакологическая группа","value":"H1-антигистаминные средства"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный"},{"name":"Минимальный возраст применения","value":"от 12 лет"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"Хранить при температуре не выше 25 °С.\u003Cbr\u003EХранить в недоступном для детей месте."},{"name":"Передозировка","value":"В исследованиях с использованием высоких доз (более 100 мг в сутки) не наблюдалось клинически значимых признаков и симптомов. Специального антидота для эбастина нет. 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При необходимости применения препарата в период лактации необходимо решить вопрос о прекращении грудного вскармливания."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"В случае возникновения побочных эффектов со стороны центральной нервной системы, таких как сонливость, необходимо соблюдать осторожность при управлении транспортными средствами и занятиях другими потенциально опасными видами деятельности, требующими повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"Эбастин может искажать результаты кожных аллергических проб. Поэтому рекомендуется проводить такие пробы не ранее, чем через 5-7 дней после отмены препарата.\u003Cbr\u003EС осторожностью:\u003Cbr\u003EПрименять у пациентов с увеличенным интервалом QT на ЭКГ, гипокалиемией, при почечной недостаточности и с легкой и умеренной степенью печеночной недостаточности (класс А, В по классификации Чайлд-Пью).\u003Cbr\u003EС осторожностью следует применять препарат Кестин при одновременном приеме с кетоконазолом или итраконазолом и эритромицином - возможно увеличение риска удлинения интервала QT на ЭКГ."},{"name":"Взаимодействие","value":"При одновременном применении препарата Кестин с кетоконазолом или итраконазолом и эритромицином возможно увеличение риска удлинения интервала QT на ЭКГ.\u003Cbr\u003EРифампицин снижает концентрацию эбастина в плазме крови и оказывает ингибирующее влияние на антигистаминный эффект эбастина.\u003Cbr\u003EПрепарат Кестин не взаимодействует с теофиллином, непрямыми антикоагулянтами, циметидином, диазепамом, этанолом и этанолсодержащими препаратами."},{"name":"Регистрационный номер","value":"ЛП-000789"},{"name":"Дата государственной регистрации","value":"14.07.2021"},{"name":"Владелец регистрационного удостоверения","value":"Almirall"},{"name":"Изготовитель","value":"Catalent U.K. Swindon Zydis Ltd"},{"name":"Фасовщик","value":"Catalent U.K. Swindon Zydis Ltd"},{"name":"Страна бренда","value":"Испания"},{"name":"Страна-производитель","value":"Великобритания"},{"name":"Название препарата","value":"Кестин"},{"name":"Срок годности","value":"36 мес."}]}],"transitionId":"tr_14979086803630941766"}}}}
Внешний вид товаров и/или упаковки может быть изменён изготовителем и отличаться от изображенных на Яндекс Маркете.

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Инструкция

Показания к применению

-аллергический ринит различной этиологии (сезонный и/или круглогодичный);
- крапивница различной этиологии, в том числе хроническая идиопатическая.

Противопоказания

- повышенная чувствительность к компонентам препарата;
- беременность;
- период лактации;
- фенилкетонурия;
- детский возраст до 12 лет;
- тяжелые нарушения функции печени (класс С по классификации Чайлд-Пью).

Способ применения и дозы

Для рассасывания в полости рта, независимо от приема пищи.
Взрослым и детям старше 12 лет рекомендуется начинать терапию с дозы 10 мг 1 раз в сутки, используя препарат Кестин, таблетки, покрытые пленочной оболочкой, 10 мг. При недостаточной эффективности или выраженной симптоматике рекомендуется использовать препарат Кестин, таблетки лиофилизированные 20 мг, по 1 таблетке 1 раз в сутки.
Курс лечения будет определяться исчезновением симптомов заболевания.
Пожилые пациенты: коррекции дозы не требуется.
Пациенты с нарушенной функцией почек: коррекции дозы не требуется. Пациенты с легкой и умеренной печеночной недостаточностью: коррекции дозы не требуется.
При тяжелых нарушениях функции печени (класс С по классификации Чайлд-Пью) суточная доза не должна превышать 10 мг, поэтому рекомендуется в этих случаях использовать препарат Кестин, таблетки, покрытые пленочной оболочкой, 10 мг.
Извлечение препарата из блистера должно осуществляться сухими руками в соответствии с инструкцией ниже:
Специальные предосторожности при обращении с препаратом:
1. Во избежание повреждения таблеток, не доставайте препарат из блистера посредством нажатия. Откройте ячейку блистера, осторожно подняв свободный край защитной пленки.
2. Снимите защитную пленку.
3. Осторожно выдавите таблетку из ячейки, не прикасаясь к ней.
4. Аккуратно извлеките препарат и положите его на язык, где он быстро растворится. Нет необходимости запивать водой или другой жидкостью, прием пищи не влияет на действие препарата.
Полная инструкция
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Кестин таб. лиоф.
Кестин таб. лиоф., 20 мг, 10 шт.
У продавца: 
нет • На Маркете: 4.8
(66)
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Инструкция
Нет в продаже
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Нет отзывов у этого продавца
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У других продавцов:66 оценок·30 отзывов
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